A Facile One Step Synthesis of 4-Aminoindoles from 5-Halo-4-oxo-4,5,6,7-tetrahydroindoles
- 1 January 1986
- journal article
- research article
- Published by The Japan Institute of Heterocyclic Chemistry in HETEROCYCLES
- Vol. 24 (6) , 1667-1674
- https://doi.org/10.3987/r-1986-06-1667
Abstract
Reaction of 5-halo-4-oxo-4,5,6,7-tetrahydroindoles with amines initiates the amination of the carbonyl function and ensuing dehydrohalogenation leads to a successful formation of 4-aminoindoles.Keywords
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