Slow antagonist dissociation and long-lasting in vivo receptor protection

• 1 July 2006
• journal article
• review article
• Published by Elsevier in Trends in Pharmacological Sciences
• Vol. 27  (7) , 355-359
• https://doi.org/10.1016/j.tips.2006.05.001

Abstract

Keywords

• DISSOCIATING ANTAGONISTS
• RECEPTOR PROTECTION
• SLOWLY DISSOCIATING
• FREE ANTAGONIST
• AGONIST CONCENTRATION
• HALF LIFE