C5-piperazinyl-1,4-benzodiazepines, water-soluble, orally bioa vailable CCKB/gastrin receptor antagonists
- 1 December 1995
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 5 (24) , 3023-3026
- https://doi.org/10.1016/0960-894x(95)00530-0
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Selective non-peptide ligands for an accommodating peptide receptor. Imidazobenzodiazepines as potent cholecystokinin type b receptor antagonistsBioorganic & Medicinal Chemistry, 1994
- Second-Generation Benzodiazepine CCK-B Antagonists. Development of Subnanomolar Analogs with Selectivity and Water SolubilityJournal of Medicinal Chemistry, 1994
- High-Affinity and Potent, Water-Soluble 5-Amino-1,4-benzodiazepine CCKB/Gastrin Receptor Antagonists Containing a Cationic Solubilizing GroupJournal of Medicinal Chemistry, 1994
- Carbamate Oxime Reduction: A New Route to C3-Amino-1,4-benzodiazepinesSynthesis, 1994
- Development of 1,4-benzodiazepine cholecystokinin type B antagonistsJournal of Medicinal Chemistry, 1993
- Molecular cloning of the human brain and gastric cholecystokinin receptor: Structure, functional expression and chromosomal localizationBiochemical and Biophysical Research Communications, 1992
- Cholecystokinin-dopamine intearctionsTrends in Pharmacological Sciences, 1991
- Effects of cholecystokinin and related peptides on neuronal activity in the ventromedial nucleus of the rat hypothalamusBritish Journal of Pharmacology, 1988
- Autoradiographic localization and biochemical characterization of peripheral type CCK receptors in rat CNS using highly selective nonpeptide CCK antagonistsJournal of Neuroscience, 1987
- Two brain cholecystokinin receptors: implications for behavioral actionsBrain Research, 1986