Synthesis, Opioid Receptor Binding, and Bioassay of Naltrindole Analogues Substituted in the Indolic Benzene Moiety

This publication has 16 references indexed in Scilit:

• Synthesis and biological evaluation of 14-alkoxymorphinans. 14.1 14-ethoxy-5-methyl substituted indolomorphinans with δ opioid receptor selectivity
  Bioorganic & Medicinal Chemistry Letters, 1997
• Effect of aromatic amino acid substitutions in the 3‐position of cyclic β‐casomorphin analogues on μ‐opioid agonist/δ‐opioid antagonist properties*
  International Journal of Peptide and Protein Research, 1996
• Attenuation of morphine tolerance and dependence with the highly selective δ-opioid receptor antagonist TIPP[ψ]
  European Journal of Pharmacology, 1995
• Electrophilic N-Benzylnaltrindoles as .delta. Opioid Receptor-Selective Antagonists
  Journal of Medicinal Chemistry, 1995
• A remarkable change of opioid receptor selectivity on the attachment of a peptidomimetic .kappa. address element to the .delta. antagonist, natrindole: 5'-[(N2-alkylamidino)methyl]naltrindole derivatives as a novel class of .kappa. opioid receptor antagonists
  Journal of Medicinal Chemistry, 1993
• Cloning of a Delta Opioid Receptor by Functional Expression
  Science, 1992
• Selective Natrexone-Derived Opioid Receptor Antagonists
  Annual Review of Pharmacology and Toxicology, 1992
• RTI-4614-4: An analog of (+)-cis-3-methylfentanyl with a 27,000-fold binding selectivity for mu versus delta opioid binding sites
  Life Sciences, 1991
• Interaction of endogenous opioid peptides and other drugs with four kappa opioid binding sites in guinea pig brain
  Peptides, 1990
• Heteroaromatic fused-ring mesoionic compounds. Sydno[3,4-a]quinoxalines
  The Journal of Organic Chemistry, 1972