Total synthesis of human cholecystokinin-33

Abstract
Human cholecystokinin (hCCK-33) has been synthesized by selective esterification of the Tyr-phenolic OH group (position 27) of unsulphated hCCK-33 with pyridine–SO3 complex after reversible masking of other functional groups by hard base (F)-labile protecting groups: amino functions by the fluoren-9-ylmethoxycarbonyl group and the Ser-OH group by the t-butyldiphenylsilyl group.

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