Asymmetric synthesis of topographically constrained amino acids: synthesis of the optically pure isomers of α,β-dimethyl-phenylalanine and α,β-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid

This publication has 11 references indexed in Scilit:

• Topographic design of peptide neurotransmitters and hormones on stable backbone templates: relation of conformation and dynamics to bioactivity
  Journal of the American Chemical Society, 1991
• Emerging approaches in the molecular design of receptor-selective peptide ligands: conformational, topographical and dynamic considerations
  Biochemical Journal, 1990
• Allylic 1,3-strain as a controlling factor in stereoselective transformations
  Chemical Reviews, 1989
• Design and synthesis of somatostatin analogs with topographical properties that lead to highly potent and specific .mu. opioid receptor antagonists with greatly reduced binding at somatostatin receptors
  Journal of Medicinal Chemistry, 1988
• Resolution and use in α-amino acid synthesis of imidazolidinone glycine derivatives
  Tetrahedron, 1988
• A new approach to receptor ligand design: synthesis and conformation of a new class of potent and highly selective μ opioid antagonists utilizing tetrahydroisoouinoline carroxylic acid
  Tetrahedron, 1988
• α‐Alkylation of Amino Acids without Racemization. Preparation of Either (S)‐ or (R)‐α‐Methyldopa from (S)‐Alanine
  Helvetica Chimica Acta, 1985
• Herstellung enantiomerenreiner cis‐ oder trans‐konfigurierter 2‐(tert‐Butyl)‐3‐methylimidazolidin‐4‐one aus den Aminosäuren (S)‐Alanin, (S)‐Phenylalanin, (R)‐Phenylglycin, (S)‐Methionin und (S)‐Valin
  Helvetica Chimica Acta, 1985
• Allylic strain in six-membered rings
  Chemical Reviews, 1968
• Über die Bildung von Isochinolin‐derivaten durch Einwirkung von Methylal auf Phenyl‐äthylamin, Phenyl‐alanin und Tyrosin
  European Journal of Inorganic Chemistry, 1911