AN EFFICIENT SYNTHESIS OF 1-ARYL-4,6-DIAMINO-1,2-DIHYDRO- 1,3,5-TRIAZINES
- 1 January 2002
- journal article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 32 (14) , 2089-2100
- https://doi.org/10.1081/scc-120005415
Abstract
1-Aryl-4,6-diamino-1,2-dihydro-1,3,5-triazines bearing diverse substituents at C2 and on the aromatic ring have been synthesized in good yield from an acid-catalyzed reaction between corresponding arylbiguanide and carbonyl compound in the presence of triethyl orthoacetate as a water scavenger.Keywords
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