Central nervous system active compounds. I. The synthesis of some caprolactam derivatives substituted at N1, C2 and C3

1 January 1976

journal article
research article
Published by CSIRO Publishing in Australian Journal of Chemistry

Vol. 29 (12) , 2651-2665
https://doi.org/10.1071/ch9762651

Abstract

The synthesis of a number of caprolactam derivatives with alkyl, aryl and hetero atom substituents at N1, C2 and C3 is described. Alkylation and arylation at C3 by a variety of methods is discussed. Some of these compounds are powerful convulsing agents; a few are depressants.

Keywords

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Central nervous system active compounds. II. The synthesis of some 4-, 5-, 6- and 7-substituted caprolactams
Australian Journal of Chemistry, 1976