Development of a model for the δ-opioid receptor pharmacophore. 4. Residue 3 dehydrophenylalanine analogues of Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13) confirm required gauche orientation of aromatic side chain
Open Access
- 6 December 1998
- journal article
- research article
- Published by Wiley in Biopolymers
- Vol. 39 (3) , 287-296
- https://doi.org/10.1002/(sici)1097-0282(199609)39:3<287::aid-bip2>3.0.co;2-k
Abstract
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This publication has 26 references indexed in Scilit:
- Development of a Model for the .delta. Opioid Receptor Pharmacophore. 1. Conformationally Restricted Tyr1 Replacements in the Cyclic .delta. Receptor Selective Tetrapeptide Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13)Journal of Medicinal Chemistry, 1994
- Conformational analysis of the .delta. receptor-selective, cyclic opioid peptide, Tyr-cyclo[D-Cys-Phe-D-Pen]OH (JOM-13). Comparison of x-ray crystallographic structures, molecular mechanics simulations, and proton NMR dataJournal of the American Chemical Society, 1994
- Validation of the general purpose QUANTA ®3.2/CHARMm® force fieldJournal of Computational Chemistry, 1992
- Synthesis, crystal structure and molecular conformation of the tBuCO‐D,L‐Ala‐Δz‐Phe‐NhiPr α,β‐unsaturated dipeptideInternational Journal of Peptide and Protein Research, 1991
- Synthesis and Molecular Structure of Stable Derivatives of (E)- and (Z)-DehydrophenylalanineAustralian Journal of Chemistry, 1991
- Conformations of dehydrophenylalanine containing peptides Nuclear Overhauser effect study of two acyclic tetrapeptidesInternational Journal of Peptide and Protein Research, 1988
- Cyclic, disulfide- and dithioether-containing opioid tetrapeptides: Development of a ligard with high delta opioid receptor selectivity and affinityLife Sciences, 1988
- Structure of an α,β-unsaturated dipeptide, racemic N-[(phenylmethoxy)carbonyl]phenylalanyl-Δ2-phenylalanineActa Crystallographica Section C Crystal Structure Communications, 1987
- Crystal structure and molecular conformation of the tripeptide, N‐Boc‐L‐Phe‐Dehydro‐Phe‐L‐Val‐OCH3Biopolymers, 1987
- Structure of ethyl (Z)-N-acetyldehydrophenylalaninate, C13H15NO3Acta Crystallographica Section C Crystal Structure Communications, 1984