A convenient method for the synthesis of macrocyclic tetra-amides by double condensation reaction

Abstract
A facile condensation reaction between bifunctional amines and carboxylic acid derivatives has been found to be very efficient for the formation of macrocyclic tetra-amide rings, and tetralactams with 33- to 37-membered rings were readily synthesized in good yields (60–90%).

This publication has 0 references indexed in Scilit: