Studies on 2-Aziridinecarboxylic Acid. VI. Synthesis of β-Alkoxy-α-Amino Acids via Ring-opening Reaction of Aziridine
- 1 September 1982
- journal article
- Published by Oxford University Press (OUP) in Bulletin of the Chemical Society of Japan
- Vol. 55 (9) , 3049-3050
- https://doi.org/10.1246/bcsj.55.3049
Abstract
The reaction of aziridine derivatives having a urethane-type protecting group with several alcohols in the presence of boron trifluoride etherate afford the corresponding optically pure O-alkylserine and O-alkylthreonine derivatives via a ring-opening reaction of aziridine in good yield.This publication has 3 references indexed in Scilit:
- Studies on 2-Aziridinecarboxylic Acid. V. Formation of Dehydroamino Acid Containing Peptides via the Isomerization by NaI of 2-Aziridinecarboxylic Acid Containing PeptidesBulletin of the Chemical Society of Japan, 1982
- Studies on 2‐aziridinecarboxylic acid peptides: Their reaction and usesBiopolymers, 1981
- Studies on Aziridine-2-carboxylic Acid. I. Synthesis of the Optically Active l-Aziridine-2-carboxylic Acid and Its DerivativesBulletin of the Chemical Society of Japan, 1978