Structure–activity relationships for 1-alkyl-3-(1-naphthoyl)indoles at the cannabinoid CB1 and CB2 receptors: steric and electronic effects of naphthoyl substituents. New highly selective CB2 receptor agonists
- 1 January 2005
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry
- Vol. 13 (1) , 89-112
- https://doi.org/10.1016/j.bmc.2004.09.050
Abstract
No abstract availableKeywords
This publication has 43 references indexed in Scilit:
- Cannabinoid receptor stimulation of guanosine-5′-O-(3-[35S]thio)triphosphate binding in rat brain membranesLife Sciences, 1996
- The two-state model of receptor activationTrends in Pharmacological Sciences, 1995
- π-π interactions: the geometry and energetics of phenylalanine-phenylalanine interactions in proteinsJournal of Molecular Biology, 1991
- Studies on a Simple Route to a Bicyclic Reserpine IntermediateSynthetic Communications, 1989
- Aromatic-Aromatic Interaction: A Mechanism of Protein Structure StabilizationScience, 1985
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973
- Photochemcial Rearrangement of N-Chloroimides to 4-Chloroimides. A New Synthesis of γ-LactonesJournal of the American Chemical Society, 1964
- The Reaction of Iodine with Some Ketones in the Presence of PyridineJournal of the American Chemical Society, 1944
- The Reaction of Furoic Acid with Aromatic Compounds*Journal of the American Chemical Society, 1941
- The Synthesis of Phenanthrene and Hydrophenanthrene Derivatives. V. The Addition of Dienes to Cyclic α,β-Unsaturated EstersJournal of the American Chemical Society, 1936