A Common Mechanism for Blockade of Heme Polymerization by Antimalarial Quinolines
Open Access
- 1 November 1998
- journal article
- Published by Elsevier in Journal of Biological Chemistry
- Vol. 273 (47) , 31103-31107
- https://doi.org/10.1074/jbc.273.47.31103
Abstract
No abstract availableKeywords
This publication has 21 references indexed in Scilit:
- An Assessment of Drug-Haematin Binding as a Mechanism for Inhibition of Haematin Polymerisation by Quinoline AntimalarialsBiochemical Pharmacology, 1998
- A Comparison and Analysis of Several Ways to Promote Haematin (Haem) Polymerisation and an Assessment of Its Initiation In VitroBiochemical Pharmacology, 1998
- HEMOGLOBIN METABOLISM IN THE MALARIA PARASITEPLASMODIUM FALCIPARUMAnnual Review of Microbiology, 1997
- Plasmodium Hemozoin Formation Mediated by Histidine-Rich ProteinsScience, 1996
- Haem polymerization in malariaNature, 1995
- Malarial haemozoin/β-haematin supports haem polymerization in the absence of proteinNature, 1995
- Quinoline anti‐malarial drugs inhibit spontaneous formation of β‐haematin (malaria pigment)FEBS Letters, 1994
- Chloroquine: Mechanism of drug action and resistance in plasmodium falciparumPharmacology & Therapeutics, 1993
- Inhibition by chloroquine of a novel haem polymerase enzyme activity in malaria trophozoitesNature, 1992
- An iron-carboxylate bond links the heme units of malaria pigment.Proceedings of the National Academy of Sciences, 1991