Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 2
- 4 October 2004
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 14 (19) , 4879-4882
- https://doi.org/10.1016/j.bmcl.2004.07.034
Abstract
No abstract availableKeywords
This publication has 12 references indexed in Scilit:
- Recent developments in the discovery of melanin-concentrating hormone antagonists: novel antiobesity agentsExpert Opinion on Therapeutic Patents, 2004
- Melanin-concentrating hormone receptor antagonists as potential antiobesity agentsExpert Opinion on Therapeutic Patents, 2002
- Rats lighten up with MCH antagonistNature Medicine, 2002
- Targeted Disruption of the Melanin-Concentrating Hormone Receptor-1 Results in Hyperphagia and Resistance to Diet-Induced ObesityEndocrinology, 2002
- T-226296: a novel, orally active and selective melanin-concentrating hormone receptor antagonistEuropean Journal of Pharmacology, 2002
- Melanin-Concentrating Hormone Receptor Is a Target of Leptin Action in the Mouse BrainEndocrinology, 2001
- Melanin-concentrating hormone overexpression in transgenic mice leads to obesity and insulin resistanceJournal of Clinical Investigation, 2001
- Melanin-concentrating Hormone Receptor: An Orphan Receptor Fits the KeyTrends in Endocrinology & Metabolism, 2000
- Mice lacking melanin-concentrating hormone are hypophagic and leanNature, 1998
- The melanin‐concentrating hormone system of the rat brain: An immuno‐ and hybridization histochemical characterizationJournal of Comparative Neurology, 1992