A novel opioid structure which accepts protonated as well as non-protonated nitrogen: A family of pure, delta receptor selective antagonists
- 1 January 1992
- journal article
- research article
- Published by Elsevier in Life Sciences
- Vol. 50 (18) , 1371-1378
- https://doi.org/10.1016/0024-3205(92)90288-z
Abstract
No abstract availableKeywords
This publication has 21 references indexed in Scilit:
- Design of peptidomimetic .delta. opioid receptor antagonists using the message-address conceptJournal of Medicinal Chemistry, 1990
- N,N-Dialkylated leucine enkephalins as potential .delta. opioid receptor antagonistsJournal of Medicinal Chemistry, 1987
- Hypophysectomy Increases TYR-MIF-1-Like Immunoreactivity in Rat PlasmaNeuroendocrinology, 1987
- Deltakephalin, Tyr-D-Thr-Gly-Phe-Leu-Thr: A new highly potent and fully specific agonist for opiate δ-receptorsBiochemical and Biophysical Research Communications, 1983
- Selective antagonists at the opiate delta-receptorLife Sciences, 1982
- Chronic ethanol imbibition interferes with δ-, but not with μ-opiate receptorsNeuropharmacology, 1981
- D‐Tyr—Ser—Gly—Phe—Leu—Thr, a highly preferential ligand for δ‐opiate receptorsFEBS Letters, 1980
- Tetrapeptide-amide analogues of enkephalin: The role of C-terminus in determining the character of opioid activityBiochemical and Biophysical Research Communications, 1979
- Endorphins are stored in biologically active and inactive forms: isolation of α-N-acetyl peptidesNature, 1979
- Differential behaviour of LPH‐(61–91)‐peptide in different model systems: Comparison of the opioid activities of LPH‐(61–91)‐peptide and its fragmentsFEBS Letters, 1977