Chiral Nonsteroidal Affinity Ligands for the Androgen Receptor. 1. Bicalutamide Analogues Bearing Electrophilic Groups in the B Aromatic Ring

This publication has 12 references indexed in Scilit:

• Affinity labeling of the androgen receptor with nonsteroidal chemoaffinity ligands
  Biochemical Pharmacology, 1999
• Discovery of Nonsteroidal Androgens
  Biochemical and Biophysical Research Communications, 1998
• Enantioselective binding of Casodex to the androgen receptor
  Xenobiotica, 1996
• Hormone binding and transcription activation by estrogen receptors: Analyses using mammalian and yeast systems
  The Journal of Steroid Biochemistry and Molecular Biology, 1993
• An androgenic affinity ligand covalently binds to cytosolic aldehyde dehydrogenase from human genital skin fibroblasts
  Molecular and Cellular Endocrinology, 1993
• Efficient and selective photoaffinity labeling of the estrogen receptor using two nonsteroidal ligands that embody aryl azide or tetrafluoroaryl azide photoreactive functions
  Biochemistry, 1991
• The Aged Rat Model of Ovarian Hormone Deficiency Bone Loss*
  Endocrinology, 1989
• Substituted 1,3,4-thiadiazoles with anticonvulsant activity. 4. Amidines
  Journal of Medicinal Chemistry, 1988
• Optimal radioligand exchange conditions for measurement of occupied androgen receptor sites in rat ventral prostate
  Archives of Biochemistry and Biophysics, 1983
• Constraints on the Flexibility of Bacteriorhodopsin's Carboxyl-Terminal Tail at the Purple Membrane Surface
  Biochemistry, 1983