Synthesis and preliminary biological evaluation of MMP inhibitor radiotracers [11C]methyl-halo-CGS 27023A analogs, new potential PET breast cancer imaging agents
- 8 October 2002
- journal article
- research article
- Published by Elsevier in Nuclear Medicine and Biology
- Vol. 29 (7) , 761-770
- https://doi.org/10.1016/s0969-8051(02)00338-4
Abstract
No abstract availableKeywords
This publication has 30 references indexed in Scilit:
- Synthesis of MMP inhibitor radiotracers [11C]methyl-CGS 27023A and its analogs, new potential PET breast cancer imaging agentsJournal of Labelled Compounds and Radiopharmaceuticals, 2002
- Potent and Selective Mechanism-Based Inhibition of GelatinasesJournal of the American Chemical Society, 2000
- Design and Synthesis of Phosphinamide-Based Hydroxamic Acids as Inhibitors of Matrix MetalloproteinasesJournal of Medicinal Chemistry, 1998
- Discovery of Potent, Achiral Matrix Metalloproteinase InhibitorsJournal of Medicinal Chemistry, 1998
- Highly Selective and Orally Active Inhibitors of Type IV Collagenase (MMP-9 and MMP-2): N-Sulfonylamino Acid DerivativesJournal of Medicinal Chemistry, 1998
- Discovery of CGS 27023A, a Non-Peptidic, Potent, and Orally Active Stromelysin Inhibitor That Blocks Cartilage Degradation in RabbitsJournal of Medicinal Chemistry, 1997
- Matrix Metalloproteinase Inhibition as a Novel Anticancer Strategy: A Review with Special Focus on Batimastat and MarimastatPharmacology & Therapeutics, 1997
- Improved synthesis of β-CIT and [11C]β-CIT labeled at nitrogen or oxygen positionsNuclear Medicine and Biology, 1996
- Stromelysin-3 expression in breast cancer biopsies: Clinico-pathological correlationsInternational Journal of Cancer, 1993
- A simple synthesis of [11C]methyl triflateInternational Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1992