Saccharin as a salt former. Enhanced solubilities of saccharinates of active pharmaceutical ingredients
- 12 January 2005
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- No. 8,p. 1073-1075
- https://doi.org/10.1039/b416137h
Abstract
Saccharin, acting as a weak acid, forms salts with basic APIs and these salts have the desirable property of enhanced water solubility.Keywords
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