Chloroethylclonidine and 2-Aminoethyl Methanethiosulfonate Recognize Two Different Conformations of the Human α2A-Adrenergic Receptor
Open Access
- 1 July 1999
- journal article
- Published by Elsevier in Journal of Biological Chemistry
- Vol. 274 (31) , 21867-21872
- https://doi.org/10.1074/jbc.274.31.21867
Abstract
No abstract availableKeywords
This publication has 26 references indexed in Scilit:
- Chloroethylclonidine Binds Irreversibly to Exposed Cysteines in the Fifth Membrane-Spanning Domain of the Human α2A-Adrenergic ReceptorMolecular Pharmacology, 1998
- Constitutive Activation of the β2 Adrenergic Receptor Alters the Orientation of Its Sixth Membrane-spanning SegmentPublished by Elsevier ,1997
- Residues in the Seventh Membrane-Spanning Segment of the Dopamine D2 Receptor Accessible in the Binding-Site CreviceBiochemistry, 1996
- Residues in the Fifth Membrane-Spanning Segment of the Dopamine D2 Receptor Exposed in the Binding-Site CreviceBiochemistry, 1995
- Recombinant human α2-adrenoceptor subtypes: comparison of [3H]rauwolscine, [3H]atipamezole and [3H]RX821002 as radioligandsBiochimica et Biophysica Acta (BBA) - Molecular Cell Research, 1995
- Mapping the binding-site crevice of the dopamine D2 receptor by the substituted-cysteine accessibility methodNeuron, 1995
- Locating ligand-binding sites in 7tm receptors by protein engineeringCurrent Opinion in Biotechnology, 1994
- Chloroethylclonidine: an irreversible agonist at prejunctional α2‐adrenoceptors in rat vas deferensBritish Journal of Pharmacology, 1993
- The cytosensor microphysiometer: biological applications of silicon technologyScience, 1992
- Molecular biology of α-adrenergic receptors: implications for receptor classification and for structure-function relationshipsBiochimica et Biophysica Acta (BBA) - Molecular Cell Research, 1991