Design and Synthesis of Novel Opiate Antagonists with LH‐Stimulating Properties
- 14 March 1990
- journal article
- research article
- Published by Wiley in Helvetica Chimica Acta
- Vol. 73 (2) , 326-336
- https://doi.org/10.1002/hlca.19900730212
Abstract
No abstract availableThis publication has 27 references indexed in Scilit:
- Crystal structures of .alpha.- and .beta.-funaltrexamine: conformational requirement of the fumaramate moiety in the irreversible blockage of .mu. opioid receptorsJournal of Medicinal Chemistry, 1986
- Multiple opioid receptor profile in vitro and activity in vivo of the potent opioid antagonist win 44,441-3Life Sciences, 1983
- Structure‐Activity Relationship of Oxygenated Morphinans. VII. 5‐Methylated and 14‐Hydroxy‐substituted Agonists and Antagonists of the 4‐Hydroxy‐ and 3, 4‐Dioxygenated 6‐Morphinanone SeriesHelvetica Chimica Acta, 1982
- Common anionic receptor site hypothesis: its relevance to the antagonist action of naloxoneJournal of Medicinal Chemistry, 1982
- Some 14.beta.-substituted analogs of N-(cyclopropylmethyl)normorphineJournal of Medicinal Chemistry, 1981
- Bremazocine: A potent, long-acting opiate kappa-agonistLife Sciences, 1980
- Relation of endogenous opioid peptides and morphine to neuroendocrine functionsLife Sciences, 1979
- 5-Allyl-9-oxobenzomorphans. 3. Potent narcotic antagonists and analgesics-antagonists in the series of substituted 2',9.beta.-dihydroxy-6,7-benzomorphansJournal of Medicinal Chemistry, 1977
- Synthesis and narcotic agonist-antagonist evaluation of some 2,6-methano-3-benzazocine-11-propanols. Analogs of the ring C bridged oripavine-7-methanolsJournal of Medicinal Chemistry, 1977
- Die Spaltung von Phenoläthern mit PyridinhydrochloridBerichte der deutschen chemischen Gesellschaft (A and B Series), 1941