Molecular Interactions of Cyclam and Bicyclam Non-peptide Antagonists with the CXCR4 Chemokine Receptor
Open Access
- 1 April 2001
- journal article
- Published by Elsevier in Journal of Biological Chemistry
- Vol. 276 (17) , 14153-14160
- https://doi.org/10.1074/jbc.m010429200
Abstract
No abstract availableKeywords
This publication has 26 references indexed in Scilit:
- Crystal Structure of Rhodopsin: A G Protein-Coupled ReceptorScience, 2000
- Phorbol Esters and SDF-1 Induce Rapid Endocytosis and Down Modulation of the Chemokine Receptor CXCR4The Journal of cell biology, 1997
- Inhibition of T-tropic HIV Strains by Selective Antagonization of the Chemokine Receptor CXCR4The Journal of Experimental Medicine, 1997
- Synthesis and Structure−Activity Relationships of Phenylenebis(methylene)- Linked Bis-tetraazamacrocycles That Inhibit Human Immunodeficiency Virus Replication. 2. Effect of Heteroaromatic Linkers on the Activity of BicyclamsJournal of Medicinal Chemistry, 1996
- Conversion of antagonist-binding site to metal-ion site in the tachykinin NK-1 receptorNature, 1995
- Synthesis and Structure-Activity Relationships of Phenylenebis(methylene)-Linked Bis-Tetraazamacrocycles That Inhibit HIV Replication. Effects of Macrocyclic Ring Size and Substituents on the Aromatic LinkerJournal of Medicinal Chemistry, 1995
- Locating ligand-binding sites in 7tm receptors by protein engineeringCurrent Opinion in Biotechnology, 1994
- Thermodynamic and kinetic data for macrocycle interactions with cations and anionsChemical Reviews, 1991
- Biosynthesis of peptide precursors and protease inhibitors using new constitutive and inducible eukaryotic expression vectorsFEBS Letters, 1990
- Site-directed mutagenesis by overlap extension using the polymerase chain reactionGene, 1989