Rs-100235: A high affinity 5-HT4 receptor antagonist
- 21 September 1995
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 5 (18) , 2119-2122
- https://doi.org/10.1016/0960-894x(95)00358-z
Abstract
No abstract availableKeywords
This publication has 9 references indexed in Scilit:
- The interaction of RS 25259‐197, a potent and selective antagonist, with 5‐HT3 receptors, in vitroBritish Journal of Pharmacology, 1995
- Synthesis and preliminary pharmacological evaluation of 2-benzyloxy substituted aryl ketones as 5-HT4 receptor antagonistsBioorganic & Medicinal Chemistry Letters, 1994
- GR113808: a novel, selective antagonist with high affinity at the 5‐HT4 receptorBritish Journal of Pharmacology, 1994
- (1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramideJournal of Medicinal Chemistry, 1993
- The 5‐HT4ReceptorMedicinal Research Reviews, 1993
- Development of a radioligand binding assay for 5‐HT4 receptors in guinea‐pig and rat brainBritish Journal of Pharmacology, 1993
- The action of SDZ 205,557 at 5‐hydroxytryptamine (5‐HT3 and 5‐HT4) receptorsBritish Journal of Pharmacology, 1993
- Mediation of 5‐hydroxytryptamine‐induced tachycardia in the pig by the putative 5‐HT4 receptorBritish Journal of Pharmacology, 1990
- Derivatives of benzo-1 : 4-dioxan. Part I. Some halogenated benzo-1 : 4-dioxans and amino- and nitro-derivatives thereofJournal of the Chemical Society, 1954