Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179)
- 9 August 2001
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 11 (18) , 2533-2536
- https://doi.org/10.1016/s0960-894x(01)00484-x
Abstract
No abstract availableKeywords
This publication has 29 references indexed in Scilit:
- Structural subtypes of the dopamine D2 receptor are functionally distinct: expression of the cloned D2A and D2B subtypes in a heterologous cell lineMolecular Endocrinology, 1992
- Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptorEuropean Journal of Pharmacology: Molecular Pharmacology, 1992
- Indole grignard reaction. III. Synthesis, crystal structure, and anglgesic activity of (R)- and (S)-3-amino-2,3,4,9-tetrahydrothiopyrano(2,3-b)indoles.CHEMICAL & PHARMACEUTICAL BULLETIN, 1990
- Synthesis of (R)-serine-2-d and its conversion to the broad-spectrum antibiotic fludalanineThe Journal of Organic Chemistry, 1987
- Access to (S)-2-methyloxetane and the precursor (S)-1,3-butanediol of high enantiomeric purityThe Journal of Organic Chemistry, 1982
- Useful syntheses of erythro- and threo-N-oleoyl-D-sphingosines (ceramides) and galactosylceramides (cerebrosides) from L-serineThe Journal of Organic Chemistry, 1981
- The reactions of an N-sulfonylamine inner saltJournal of the American Chemical Society, 1968
- Elaiomycin. II. Determination of the D-threo ConfigurationJournal of the American Chemical Society, 1959
- 126. The stereochemistry of an oxazoline derivative of threonine. Improvement of a recent threonine synthesisJournal of the Chemical Society, 1949
- Aryloxyacetamidines and 2-(Aryloxymethyl)-imidazolines1Journal of the American Chemical Society, 1947