Synthesis, biochemical and pharmacological properties of BUBUC, a highly selective and systemically active agonist for in vivo studies of δ-opioid receptors

This publication has 39 references indexed in Scilit:

• Tritium labelling of highly selective probes for δ‐opioid receptors: [³H] Tyr‐D‐Ser(O‐t‐Bu)‐Gly‐Phe‐Leu‐Thr(DSTBULET) and [³H]Tyr‐D‐Ser(O‐t‐Bu)‐Gly‐Phe‐Leu‐Thr(O‐t‐Bu)(BUBU)
  Journal of Labelled Compounds and Radiopharmaceuticals, 1990
• Isolation of dermenkephalin from amphibian skin, a high‐affinity (δ‐selective opioid heptapeptide containing a D‐amino acid residue
  FEBS Letters, 1989
• .delta. Opioid receptor selectivity induced by conformational constraints in linear enkephalin-related peptides: proton 400-MHz NMR study and theoretical calculations
  Biochemistry, 1989
• Can supraspinal δ-opioid receptors mediate antinociception?
  Trends in Pharmacological Sciences, 1988
• The Physiology and Pharmacology of Spinal Opiates
  Annual Review of Pharmacology and Toxicology, 1985
• INTRATHECAL DELTA-RECEPTOR LIGAND PRODUCES ANALGESIA IN MAN
  The Lancet, 1983
• Deltakephalin, Tyr-D-Thr-Gly-Phe-Leu-Thr: A new highly potent and fully specific agonist for opiate δ-receptors
  Biochemical and Biophysical Research Communications, 1983
• Analgesic activity of intracerebroventricular administration of morphiceptin and β-casomorphins: Correlation with the morphine (μ) receptor binding affinity
  Life Sciences, 1982
• D‐Tyr—Ser—Gly—Phe—Leu—Thr, a highly preferential ligand for δ‐opiate receptors
  FEBS Letters, 1980
• Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
  Biochemical Pharmacology, 1973