Design and Synthesis of 1,4-Diazabicyclo[4.3.0]nonane Peptidomimetic Endothelin Antagonists

This publication has 13 references indexed in Scilit:

• Discovery of endothelin antagonists
  Published by Walter de Gruyter GmbH ,1997
• Structure-Activity Relationships of Cyclic Pentapeptide Endothelin A Receptor Antagonists
  Journal of Medicinal Chemistry, 1995
• Solvent effects on the conformation of cyclo(‐D‐Trp‐D‐Asp‐Pro‐D‐val‐Leu‐) An NMR spectroscopy and molecular modeling study
  International Journal of Peptide and Protein Research, 1994
• Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor
  Life Sciences, 1992
• The solution structure of a cyclic endothelin antagonist, BQ‐123, based on¹H–¹H and¹³H–¹H three bond oupling constants
  FEBS Letters, 1992
• Solution conformation of a cyclic pentapeptide endothelin antagonist Comparison of structures obtained from constrained dynamics and conformational search
  FEBS Letters, 1992
• Conformational study of cyclo[D‐Trp‐D‐Asp‐Pro‐D‐Val‐Leu], an endothelin‐A receptor‐selective antagonist
  FEBS Letters, 1992
• A novel potent vasoconstrictor peptide produced by vascular endothelial cells
  Nature, 1988
• Oxidation of long-chain and related alcohols to carbonyls by dimethyl sulfoxide "activated" by oxalyl chloride
  The Journal of Organic Chemistry, 1978
• Bicyclic Homologs of Piperazine. Synthesis of 8-Methyl-3,8-diazabicyclooctanes. I
  The Journal of Organic Chemistry, 1961