Preparation of 2,4‐diamino‐6‐(diallylamino)‐s‐triazine‐2,4‐14c and its hypotensive metabolite, 2,4‐diamino‐6‐(diallylamino)‐s‐triazine‐2,4‐14c 3‐oxide
- 1 January 1978
- journal article
- research article
- Published by Wiley in Journal of Labelled Compounds and Radiopharmaceuticals
- Vol. 14 (6) , 807-811
- https://doi.org/10.1002/jlcr.2580140603
Abstract
2,4‐Diamino‐6‐(diallylamino)‐s‐triazine‐2,4‐14C was prepared from K14CN in a four step sequence of reactions. The product was obtained in 26% yield at a specific activity of 1.01 mCi per mM. This product was converted to the hypotensive agent, 2,4‐diamino‐6‐(diallylamino)‐s‐triazine‐2,4‐14C 3‐oxide in 37% yield by oxidation with m‐chloroperbenzoic acid.Keywords
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