Oximino-piperidino-piperidine-based CCR5 antagonists. Part 2: synthesis, SAR and biological evaluation of symmetrical heteroaryl carboxamides
- 1 February 2003
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 13 (4) , 709-712
- https://doi.org/10.1016/s0960-894x(02)01063-6
Abstract
No abstract availableKeywords
This publication has 20 references indexed in Scilit:
- Small molecule antagonists of chemokine receptors as emerging anti-HIV agentsExpert Opinion on Therapeutic Patents, 2001
- CHEMOKINE RECEPTORS AS HIV-1 CORECEPTORS: Roles in Viral Entry, Tropism, and DiseaseAnnual Review of Immunology, 1999
- Chemokine Receptors: Keys to AIDS Pathogenesis?Cell, 1998
- Resistance to HIV-1 infection in Caucasian individuals bearing mutant alleles of the CCR-5 chemokine receptor geneNature, 1996
- Homozygous Defect in HIV-1 Coreceptor Accounts for Resistance of Some Multiply-Exposed Individuals to HIV-1 InfectionCell, 1996
- Identification of RANTES, MIP-1α, and MIP-1β as the Major HIV-Suppressive Factors Produced by CD8 + T CellsScience, 1995
- Synthesis and Proton Nmr Spectra of the Monomethyl- and dimethylpyrimidine-5-carboxylic Acids. Regioselective Covalent Hydration at the 2- and 4-Ring PositionsHETEROCYCLES, 1994
- Procedures for the acylation of diethyl malonate and ethyl acetoacetate with acid chlorides using tertiary amine bases and magnesium chlorideThe Journal of Organic Chemistry, 1985
- Reaction of N-Aminopyridinium Derivatives. V. Syntheses of 1-(N-Methylacetamido) alkylpyridinium Salts and Their Reaction with Cyanide Ion.CHEMICAL & PHARMACEUTICAL BULLETIN, 1966
- Synthese substituierter Hydrazine aus Aminen mit Hydroxylamin‐O‐sulfonsäureEuropean Journal of Inorganic Chemistry, 1959