Evidence for low brain penetration by the H1-receptor antagonist temelastine (SK & F 93944)
- 1 January 1987
- journal article
- research article
- Published by Elsevier in European Journal of Pharmacology
- Vol. 133 (1) , 65-74
- https://doi.org/10.1016/0014-2999(87)90206-8
Abstract
No abstract availableKeywords
This publication has 15 references indexed in Scilit:
- Pharmacological studies with SK&F 93944 (temelastine), a novel histamine H1‐receptor antagonist with negligible ability to penetrate the central nervous systemBritish Journal of Pharmacology, 1986
- HISTAMINE H1‐AGONIST POTENTIATION OF ADENOSINE‐STIMULATED CYCLIC AMP ACCUMULATION IN SLICES OF GUINEA‐PIG CEREBRAL CORTEX: COMPARISON OF RESPONSE AND BINDING PARAMETERSBritish Journal of Pharmacology, 1982
- Antihistaminic effect of terfenadine: A new piperidine-type antihistamineDrug Development Research, 1982
- Effect of mequitazine a non sedative antihistamine on brain H1 receptorsLife Sciences, 1981
- Histamine H1-receptors labeled in vivo: Antidepressant and antihistamine interactionsEuropean Journal of Pharmacology, 1980
- Neurotransmitter Receptor Binding in Bovine Cerebral MicrovesselsScience, 1980
- HISTAMINE H1‐RECEPTORS IN THE BRAIN OF THE GUINEA‐PIG AND THE RAT: DIFFERENCES IN LIGAND BINDING PROPERTIES AND REGIONAL DISTRIBUTIONBritish Journal of Pharmacology, 1980
- HETEROGENEITY OF HISTAMINE Hi‐RECEPTORS: SPECIES VARIATIONS IN [3H]MEPYRAMINE BINDING OF BRAIN MEMBRANESJournal of Neurochemistry, 1979
- THE BINDING OF [3H]MEPYRAMINE TO HISTAMINE H1 RECEPTORS IN GUINEA‐PIG BRAINJournal of Neurochemistry, 1978
- Studies on the effects of histaminergic agents on seizure susceptibility in micePsychopharmacology, 1976