Novel enantioselective acylating agents. The reactions of chiral ortho esters and silylenol ethers as a route to optically active monoprotected 1,3-dicarbonyl compounds

Abstract
A novel enantioselective route to monoprotected 2-substituted-1,3-dicarbonyl compounds has been developed via acylation of silylenol ethers with chiral ortho esters derived from diethyl or di-isopropyl (R,R)-tartrates; good yields and stereoselectivity can be achieved starting from cyclic enolsilanes.

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