Aryl–aryl coupling via directed lithiation and oxidation
- 12 April 2005
- journal article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- No. 20,p. 2589-2590
- https://doi.org/10.1039/b501939g
Abstract
Aryl lithium reagents formed by directed lithiation reactions undergo transmetallation with copper(I) salts to form organocuprates, which may be efficiently oxidized to yield ortho-substituted biaryls.Keywords
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