Synthesis of SB-214857 using Copper Catalysed Amination of Arylbromides with l-Aspartic Acid
- 28 August 2001
- journal article
- letter
- Published by Georg Thieme Verlag KG in Synlett
- Vol. 2001 (09) , 1423-1427
- https://doi.org/10.1055/s-2001-16780
Abstract
An efficient synthesis of a 1,4-benzodiazepine was accomplished using copper catalysed amination of an arylbromide with the soluble bis-tetrabutylammonium salt of l-aspartic acid as a key step.Keywords
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