Development of 123I-labelled NNC 13-8241 as a radioligand for SPECT visualization of benzodiazepine receptor binding
- 1 April 1996
- journal article
- Published by Elsevier in Nuclear Medicine and Biology
- Vol. 23 (3) , 201-209
- https://doi.org/10.1016/0969-8051(95)02041-1
Abstract
No abstract availableKeywords
This publication has 19 references indexed in Scilit:
- Radioligands for PET studies of central benzodiazepine receptors and PK (peripheral benzodiazepine) binding sites—current statusNuclear Medicine and Biology, 1993
- Neuroreceptor Quantitation in vivo by the Steady-State Principle Using Constant Infusion or Bolus Injection of Radioactive TracersJournal of Cerebral Blood Flow & Metabolism, 1992
- Receptor binding characterization of the benzodiazepine radioligand 125I-Ro16-0154: Potential probe for spect brain imagingLife Sciences, 1990
- Metabolism of the benzodiazepine antagonist11C-Ro 15-1788 after intravenous administration in manHuman Psychopharmacology: Clinical and Experimental, 1989
- Cerebral uptake of 11C—Ro 15—1788 and its acid metabolite 11C—Ro 15—3890; PET study in healthy volunteersHuman Psychopharmacology: Clinical and Experimental, 1989
- 11C-labelling of Ro 15-1788 in two different positions, and also 11C-labelling of its main metabolite Ro 15-3890, for PET studies of benzodiazepine receptorsInternational Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1988
- Synthesis of ethyl 8-fluoro-5,6-dihydro5- [11C]methyl-6-oxo-4H-imidazo[1,5-a] [1,4]benzodiazepine-3-carboxylate (RO 15.1788-11C): A specific radioligand for the in vivo study of central benzodiazepine receptors by positron emission tomographyThe International Journal of Applied Radiation and Isotopes, 1984
- Central type benzodiazepine binding sites: A positron emission tomography study in the baboon's brainNeuroscience Letters, 1984
- Radioiodination techniques for small organic moleculesChemical Reviews, 1982
- Position-specific radioiodination utilizing an aryltributylstannyl intermediate. Synthesis of 125I-iodotamoxifenThe International Journal of Applied Radiation and Isotopes, 1981