SYNTHESIS and STRUCTURE-ACTIVITY RELATIONSHIPS in PERHYDROISOINDOLE SUBSTANCE P ANTAGONISTS
- 1 January 1995
- journal article
- Published by Elsevier in European Journal of Medicinal Chemistry
- Vol. 30, 575s-585s
- https://doi.org/10.1016/s0223-5234(23)00152-6
Abstract
No abstract availableThis publication has 26 references indexed in Scilit:
- Synthesis of RPR 100893, prototype of a new series of potent and selective non peptide NK1 antagonists : the triarylperhydroisoindolols.Bioorganic & Medicinal Chemistry Letters, 1994
- Perhydrothiopyranopyrroles derivatives : A novel series of potent and selective nonpeptide NK1 antagonists.Bioorganic & Medicinal Chemistry Letters, 1994
- Patent Update: Neurokinin Receptor AntagonistsCurrent Opinion on Therapeutic Patents, 1993
- Tachykinin receptors and tachykinin receptor antagonistsJournal of Autonomic Pharmacology, 1993
- Synthesis of RP-67,580, a new potent nonpeptide substance P antagonistBioorganic & Medicinal Chemistry Letters, 1992
- Toward nonpeptidal substance P mimetic analogues: Design, synthesis, and biological activityBiopolymers, 1991
- Modulation of neurogenic inflammation: novel approaches to inflammatory diseaseTrends in Pharmacological Sciences, 1990
- New selective agonists for neurokinin receptors: pharmacological tools for receptor characterizationTrends in Pharmacological Sciences, 1988
- Does substance P act as a pain transmitter?Trends in Pharmacological Sciences, 1987
- N-(TRIMETHYLSILYLMETHYL)AMINOMETHYL ETHERS AS AZOMETHINE YLIDE SYNTHONS. A NEW AND CONVENIENT ACCESS TO PYRROLIDINE DERIVATIVESChemistry Letters, 1984