An Efficient Fischer Indole Synthesis of Avitriptan, a Potent 5-HT_1D Receptor Agonist

This publication has 14 references indexed in Scilit:

• Effects of avitriptan, a new 5-HT1B/1D receptor agonist, in experimental models predictive of antimigraine activity and coronary side-effect potential
  Naunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie, 1997
• 4-Hydroxy-2-methyl-3(2H)-isothiazolone-1,1-dioxide as protecting group of 4-(N-methylaminosulfonyl)methylphenylhydrazine during Fischer indole synthesis
  Tetrahedron Letters, 1995
• MK-0462
  Drugs of the Future, 1995
• Improved Fischer Indole Reaction for the Preparation of N,N-Dimethyltryptamines: Synthesis of L-695,894, a Potent 5-HT1D Receptor Agonist
  The Journal of Organic Chemistry, 1994
• The synthesis of a conformationally restricted analog of the anti-migraine drug sumatriptan
  Tetrahedron Letters, 1992
• Fluticasone propionate
  Drugs of Today, 1992
• Synthesis of indoles via palladium-catalyzed heteroannulation of internal alkynes
  Journal of the American Chemical Society, 1991
• A Novel Approach to the Synthesis of 7(Z), 11(Z)-Nonacosadiene, Pheromone of Drosophila Melano Gaster and 9(Z)-Tricosene, Pheromone of Musca Domestica
  Synthetic Communications, 1989
• Fast and selective oxidation of primary alcohols to aldehydes or to carboxylic acids and of secondary alcohols to ketones mediated by oxoammonium salts under two-phase conditions
  The Journal of Organic Chemistry, 1987
• Cleavage of Cyclic Ethers with Boron Bromide. A Convenient Route to the Bromosubstituted Alcohols, Aldehydes and Ketones
  HETEROCYCLES, 1982