Mutational analysis of the putative devazepide binding site of the CCKA receptor

This publication has 16 references indexed in Scilit:

• Recovery from TPA inhibition of receptor-mediated Ca2+ mobilization is paralleled by down-regulation of protein kinase C-α in CHO cells expressing the CCK-A receptor
  Cell Calcium, 1996
• His381 of the rat CCKB receptor is essential for CCKB versus CCKA receptor antagonist selectivity
  European Journal of Pharmacology, 1996
• The role of the Val353 residue in antagonist binding to rat CCK-B receptors
  NeuroReport, 1995
• The Role of the Cholecystokinin-B/Gastrin Receptor Transmembrane Domains in Determining Affinity for Subtype-selective Ligands(∗)
  Published by Elsevier ,1995
• A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists
  Nature, 1993
• Chemical modification of cholecystokinin‐A receptors in rat pancreatic membranes
  European Journal of Biochemistry, 1992
• Cholecystokinin receptors: synthetic antagonists with selectivity for receptor subtypes and possible clinical applications
  Biochemical Society Transactions, 1991
• Effects of a novel cholecystokinin (CCK) receptor antagonist, MK-329, on gallbladder contraction and gastric emptying in humans. Implications for the physiology of CCK.
  Journal of Clinical Investigation, 1989
• ROLE OF CHOLECYSTOKININ IN REGULATION OF GASTROINTESTINAL MOTOR FUNCTIONS
  The Lancet, 1989
• Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists
  Journal of Medicinal Chemistry, 1988