Structure-activity relationships within a series of analogues of the histamine H1-antagonist terfenadine
- 1 January 1993
- journal article
- Published by Elsevier in European Journal of Medicinal Chemistry
- Vol. 28 (2) , 165-173
- https://doi.org/10.1016/0223-5234(93)90009-4
Abstract
No abstract availableKeywords
This publication has 13 references indexed in Scilit:
- Comparative study of central and peripheral histamine-H1 receptor binding in vitro and ex vivo of non-sedating antihistamines and of noberastine, a new agentDrug Development Research, 1991
- Enantiomeric analysis of terfenadine in rat plasma by HPLCChirality, 1991
- TerfenadineDrugs, 1990
- Synthesis of alkyl-substituted N-protected indoles via acylation and reductive deoxygenationThe Journal of Organic Chemistry, 1989
- Synthesis and antiallergy activity of 4-(diarylhydroxymethyl)-1-[3-(aryloxy)propyl)piperidines and structurally related compoundsJournal of Medicinal Chemistry, 1989
- Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonistsJournal of Medicinal Chemistry, 1988
- Chiral synthesis via organoboranes. 14. Selective reductions. 41. Diisopinocampheylchloroborane, an exceptionally efficient chiral reducing agentJournal of the American Chemical Society, 1988
- 2-Chloro-4(R),5(R)-dimethyl-2-oxo-1,3,2-dioxaphospholane, a new chiral derivatizing agentThe Journal of Organic Chemistry, 1984
- Reactions of Sodium Borohydride in Acidic Media; VII. Reduction of Diaryl Ketones in Trifluoroacetic AcidSynthesis, 1978
- Nitramine; III1. Alkylthiomethyl- und Arylthiomethyl-nitramine und ihre SulfoneSynthesis, 1973