A Convenient Route to Condensed-Ring Aromatic Acetylenes
- 1 July 1998
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 28 (14) , 2571-2576
- https://doi.org/10.1080/00397919808004825
Abstract
Palladium catalysed coupling of aryl halides with 3-methylbut-1-yn-3-ol and a subsequent base-induced retro-Favorsky reaction gave the corresponding ethynyl aromatics in good to excellent yields.Keywords
This publication has 16 references indexed in Scilit:
- Preparation of sterically constrained arylalkynesTetrahedron, 1997
- Preparation of sterically constrained arylalkyne oligomersTetrahedron, 1997
- Synthesis of 1,4-di(n-pyridyl)buta-1,3-diyne and formation of charge-transfer complexes. X-Ray structure of 1,4-di(3-pyridyl)buta-1,3-diyneJournal of the Chemical Society, Perkin Transactions 1, 1997
- Mechanism-based inhibition of mouse P4502b-10 by selected arylalkynesBiochemical Pharmacology, 1996
- Synthesis and chiroptical properties of axially chiral, binaphthol-based oligomersTetrahedron Letters, 1996
- Interaction of 1-ethynylpyrene and hepatic CYPIA1 from rainbow troutChemico-Biological Interactions, 1994
- Synthesis and 5-Lipoxygenase Inhibitory Activities of Some Novel 2-Substituted 5-Benzofuran Hydroxamic AcidsJournal of Medicinal Chemistry, 1994
- Determinants of protein modification versus heme alkylation: inactivation of cytochrome P450 1A1 by 1-ethynylpyrene and phenylacetyleneChemical Research in Toxicology, 1993
- Suicide inhibitors of cytochrome P450 1A1 and P450 2B1Biochemical Pharmacology, 1992
- Linear Conjugated Systems Bearing Aromatic Terminal Groups. V. Syntheses and Electronic Spectra of 2,2′-, 3,3′-, and 9,9′-Diphenanthrylpoly-ynesBulletin of the Chemical Society of Japan, 1971