The synthesis and opioid receptor binding affinities of analogues of dermorphin and its N-terminal tetrapeptide fragment with dibasic acids in position 2
- 22 September 1995
- journal article
- Published by Elsevier in Life Sciences
- Vol. 57 (18) , 1633-1640
- https://doi.org/10.1016/0024-3205(95)02142-6
Abstract
No abstract availableKeywords
This publication has 20 references indexed in Scilit:
- Design of cyclic deltorphins and dermenkephalins with a disulfide bridge leads to analogs with high selectivity for .delta.-opioid receptorsJournal of Medicinal Chemistry, 1994
- Cyclic enkephalin analogs with exceptional potency at peripheral .delta. opioid receptorsJournal of Medicinal Chemistry, 1994
- Topographical requirements for delta opioid ligands: Common structural features of dermenkephalin and deltorphinLife Sciences, 1992
- Topographical requirements for delta opioid ligands: Presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activityBiochemical and Biophysical Research Communications, 1991
- Dermorphin analogs carrying an increased positive net charge in their "message" domain display extremely high .mu.-opioid receptor selectivityJournal of Medicinal Chemistry, 1989
- A high affinity, highly selective ligand for the delta opioid receptor: [3H]-[D-PEN2, pCl-PHE4, D-PEN5]enkephalinLife Sciences, 1989
- PCNONLIN and NONLIN84: Software for the Statistical Analysis of Nonlinear ModelsThe American Statistician, 1986
- A comparison of the antinociceptive and behavioral effects of D-Arg substituted dipeptides and tetrapeptides in micePeptides, 1985
- Opioid activity of enkephalin analogues containing the kyotorphin-related structure in the N-terminusNeuropharmacology, 1984
- AMINO ACID COMPOSITION AND SEQUENCE OF DERMORPHIN, A NOVEL OPIATE‐LIKE PEPTIDE FROM THE SKIN OF PHYLLOMEDUSA SAUVAGEIInternational Journal of Peptide and Protein Research, 1981