How to increase the reactivity of [18F]fluoroethyl bromide: [18F]fluoroethylation of amine, phenol and amide functional groups with [18F]FEtBr, [18F]FEtBr/NaI and [18F]FEtOTf

This publication has 16 references indexed in Scilit:

• Synthesis and preliminary PET study of the 5‐HT₇ receptor antagonist [¹¹C]DR4446
  Journal of Labelled Compounds and Radiopharmaceuticals, 2002
• N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: A Potent and Selective Dopamine D₄ Ligand
  Journal of Medicinal Chemistry, 1998
• Radiosynthesis and biodistribution of the S-[18F]fluoroethyl analog of McN5652
  Nuclear Medicine and Biology, 1996
• Pet imaging studies of dopamine D₂ receptors: Comparison of [¹⁸F]N‐Methylspiperone; and the benzamide analogues [¹⁸F]MABN and [¹⁸F]MBP in baboon brain
  Synapse, 1995
• Improved synthesis of some commonly used PET radioligands by the use of [11C]methyl triflate
  Nuclear Medicine and Biology, 1995
• A simple synthesis of [11C]methyl triflate
  International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1992
• A rapid and efficient method for the fluoroalkylation of amines and amides. Development of a method suitable for incorporation of the short-lived positron emitting radionuclide fluorine-18
  The Journal of Organic Chemistry, 1987
• Synthesis of no-carrier-added N-([18F]fluoroalkyl)spiperone derivatives
  International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1986
• Quantitative Analysis of D2 Dopamine Receptor Binding in the Living Human Brain by PET
  Science, 1986
• Syntheses and D2 receptor affinities of derivatives of spiperone containing aliphatic halogens
  Applied Radiation and Isotopes, 1986