Structure-activity relationships of enkephalins containing serially replaced thiomethylene amide bond surrogates
- 1 April 1986
- journal article
- research article
- Published by Elsevier in Life Sciences
- Vol. 38 (14) , 1243-1249
- https://doi.org/10.1016/0024-3205(86)90416-9
Abstract
No abstract availableThis publication has 16 references indexed in Scilit:
- Enkephalin pseudopeptides: Resistance to in vitro proteolytic degradation afforded by amide bond replacements extends to remote sitesPeptides, 1985
- Evidence of a peptide backbone contribution toward selective receptor recognition for leucine enkephalin thioamide analogsBiochemical and Biophysical Research Communications, 1984
- Replacement of the peptide-backbone amides connecting Tyr-Gly and Gly-Gly in leucine-enkephalin with ketomethylene groups: synthesis and biological activityJournal of Medicinal Chemistry, 1984
- Selective antagonists at the opiate delta-receptorLife Sciences, 1982
- Conformational restrictions of biologically active peptides via amino acid side chain groupsLife Sciences, 1982
- On the double bond isostere of the peptide bond: preparation of an enkephalin analogueJournal of the Chemical Society, Perkin Transactions 1, 1982
- Synthesis and biological activities of pseudopeptide analogues of LH-RH: Agonists and antagonistsBiochemical and Biophysical Research Communications, 1980
- METHIONINE ENKEPHALIN AND ISOSTERIC ANALOGUESInternational Journal of Peptide and Protein Research, 1980
- Incorporation of trans-olefinic dipeptide isosteres into enkephalin and substance P analoguesJournal of the Chemical Society, Chemical Communications, 1980
- Synthesis of oxytocin and related diastereomers deuterated in the half-cystine positions. Comparison of solid-phase and solution methodsThe Journal of Organic Chemistry, 1974