Synthesis of Constrained Raloxifene Analogues by Complementary Use of Friedel−Crafts and Directed Remote Metalation Reactions
- 28 June 2003
- journal article
- research article
- Published by American Chemical Society (ACS) in The Journal of Organic Chemistry
- Vol. 68 (15) , 5992-5999
- https://doi.org/10.1021/jo034325k
Abstract
No abstract availableKeywords
This publication has 15 references indexed in Scilit:
- Cross-coupling reactions via organoboranesJournal of Organometallic Chemistry, 2002
- Hormone replacement therapy and cardiovascular diseaseCurrent Opinion in Lipidology, 1999
- Synthesis and Pharmacology of Conformationally Restricted Raloxifene Analogues: Highly Potent Selective Estrogen Receptor ModulatorsJournal of Medicinal Chemistry, 1998
- Structure−Activity Relationships of Selective Estrogen Receptor Modulators: Modifications to the 2-Arylbenzothiophene Core of RaloxifeneJournal of Medicinal Chemistry, 1997
- Destabilized carbocations. Nuclear magnetic resonance detection and reactivities of aryl α-thioformamidyl cationsCanadian Journal of Chemistry, 1987
- Rapid removal of protecting groups from peptides by catalytic transfer hydrogenation with 1,4-cyclohexadieneThe Journal of Organic Chemistry, 1978
- B-bromo-9-borabicyclo[3.3.1]nonane. A convenient and selective reagent for ether cleavageJournal of Organometallic Chemistry, 1978
- Thianaphthen-2-one chemistry. 2. The benzylidene thiolactone rearrangement: synthesis of 2-arylthianaphthene-3-carboxylic acids and estersThe Journal of Organic Chemistry, 1976
- Thianaphthen-2-one chemistry. I. Synthesis of 6H-benzothieno[3,2-c][1]benzopyran-6-ones (11-thiacoumestans)The Journal of Organic Chemistry, 1975
- 4-Morpholinomethyl Alkyl Ethers and N-Substituted MorpholinesJournal of the American Chemical Society, 1940