A High-Content Glucocorticoid Receptor Translocation Assay for Compound Mechanism-of-Action Evaluation
Open Access
- 1 December 2007
- journal article
- other
- Published by Elsevier in SLAS Discovery
- Vol. 12 (8) , 1029-1041
- https://doi.org/10.1177/1087057107309353
Abstract
No abstract availableKeywords
This publication has 51 references indexed in Scilit:
- Dissociated non-steroidal glucocorticoids: tuning out untoward effectsExpert Opinion on Therapeutic Patents, 2007
- Controlling nuclear receptors: the circular logic of cofactor cyclesNature Reviews Molecular Cell Biology, 2005
- Coactivators in Assay Design for Nuclear Hormone Receptor Drug DiscoveryASSAY and Drug Development Technologies, 2003
- Multiplexing Nuclear Receptors for Agonist Identification in a Cell-Based Reporter Gene High-Throughput ScreenSLAS Discovery, 2003
- A Comparison of ALPHAScreen, TR-FRET, and TRF as Assay Methods for FXR Nuclear ReceptorsSLAS Discovery, 2002
- A High-Throughput Fluorescent Polarization Assay for Nuclear Receptor Binding Utilizing Crude Receptor ExtractAnalytical Biochemistry, 2002
- Use of Homogeneous Time-Resolved Fluorescence Energy Transfer in the Measurement of Nuclear Receptor ActivationMethods, 2001
- Development of High Throughput Screening Assays Using Fluorescence Polarization: Nuclear Receptor-Ligand–Binding and Kinase /Phosphatase AssaysSLAS Discovery, 2000
- Green fluorescent protein (GFP): applications in cell-based assays for drug discoveryDrug Discovery Today, 1999
- The nuclear receptor superfamily: The second decadeCell, 1995