A brief study of the selectivity of norbinaltorphimine, (−)-cyclofoxy, and (+)-cyclofoxy among opioid receptor subtypes in vitro
- 1 October 1988
- journal article
- research article
- Published by Elsevier in Neuropeptides
- Vol. 12 (3) , 181-187
- https://doi.org/10.1016/0143-4179(88)90052-2
Abstract
No abstract availableThis publication has 19 references indexed in Scilit:
- Binaltorphimine-related bivalent ligands and their .kappa. opioid receptor antagonist selectivityJournal of Medicinal Chemistry, 1988
- LY164929: a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding siteNeuropeptides, 1988
- Tritiated-6-beta-fluoro-6-desoxy-oxymorphone 〈[3H] FOXY〉: a new ligand and photoaffinity probe for the MU opioid receptorsNeuropeptides, 1988
- Chronic morphine upregulates a μ-opiate binding site labeled by [3H]cycloFOXY: a novel opiate antagonist suitable for positron emission tomographyEuropean Journal of Pharmacology, 1987
- Binaltorphimine and nor-binaltorphimine, potent and selective k-opioid receptor antagonistsLife Sciences, 1987
- Preparation of rat brain membranes highly enriched with opiate kappa binding sites using site-directed acylating agents: Optimization of assay conditionsNeuropeptides, 1985
- S‐[18F]Acetylcyclofoxy: a useful probe for the visualization of opiate receptors in living animalsFEBS Letters, 1984
- Preparation of rat brain membranes greatly enriched with either type-I-delta or type-II-delta opiate binding sites using site directed alkylating agents: Evidence for a two-site allosteric modelNeuropeptides, 1984
- Binding of radiolabeled opiates to slide-mounted sections of molded minced rat brain: A novel method for conducting radioreceptor assaysNeuropeptides, 1983
- Irreversible Ligands with High Selectivity Toward δ and μ Opiate ReceptorsScience, 1983