Two Simple Methods for the Synthesis of Trialkyl ?-Aminophosphono-Acetates ( 3 ). Trifluoromethanesulfonyl Azide as an Azide-Transfer Agent
- 1 January 1980
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 10 (6) , 429-435
- https://doi.org/10.1080/00397918008064265
Abstract
In connection with a cephalosporin synthesis,1 Ratcliffe and Christensen reported the preparation of alkyl α-aminodiethylphos-phonoacetate2 3. We experienced considerable difficulty in repeating the procedure reported, and wish to describe alternate simple, high-yield preparations of 3.Keywords
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