Application of the Intramolecular α-Amidoalkylation Reaction for the Synthesis of 3- and 1,3-Alkyl(aryl) 2-Formyltetrahydroisoquinolines
- 1 June 1993
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 23 (12) , 1707-1719
- https://doi.org/10.1080/00397919308011269
Abstract
3- and 1,3-Alkyl(aryl) 2-Formyltetrahydroisoquinolines 6 are obtained by the application of the intramolecular α-amidoalkylation reaction from 1-Alkyl(Aryl) 2-Arylethy1formamides 2 and aldehydes in acidic medium.Keywords
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