Potency and selectivity of the tachykinin NK3 receptor antagonist SR142801

This publication has 28 references indexed in Scilit:

• Neurokinin A (NK2) receptor revisited with SR 48968, a potent non-peptide antagonist
  Published by Elsevier ,2005
• The 'septide-sensitive' tachykinin receptor: still an enigma
  Trends in Pharmacological Sciences, 1995
• SR 142801, The first potent non-peptide antagonist of the tachykinin NK3 receptor
  Life Sciences, 1994
• The Nonpeptide Tachykinin NK2 Receptor Antagonist SR 48968 Interacts with Human, but Not Rat, Cloned Tachykinin NK3 Receptors
  Biochemical and Biophysical Research Communications, 1994
• Molecular characterisation, expression and localisation of human neurokinin‐3 receptor
  FEBS Letters, 1992
• Phylogeny of tachykinin receptor localization in the vertebrate central nervous system: apparent absence of neurokinin-2 and neurokinin-3 binding sites in the human brain
  Brain Research, 1991
• Neurokinin3-receptors are linked to inositol phospholipid hydrolysis in the guinea-pig ileum longitudinal muscle-myenteric plexus preparation
  British Journal of Pharmacology, 1988
• Effects of tachykinins on inositol phospholipid hydrolysis in slices of hamster urinary bladder
  British Journal of Pharmacology, 1987
• Multiple tachykinin binding sites in hamster, rat and guinea-pig urinary bladder
  European Journal of Pharmacology, 1986
• Homocysteine thiolactone as precursor of methionine amide : application to the modification of peptides of the tachykinin family
  Tetrahedron Letters, 1985