Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin‐like activity
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Open Access
- 9 October 2000
- journal article
- Published by Wiley in FEBS Letters
- Vol. 483 (1) , 52-56
- https://doi.org/10.1016/s0014-5793(00)02082-2
Abstract
Some synthetic agonists of the VR1 vanilloid (capsaicin) receptor also inhibit the facilitated transport into cells of the endogenous cannabinoid anandamide (arachidonoylethanolamide, AEA). Here we t...Keywords
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