Asymmetric Synthesis of Both Enantiomers of α-Trifluoromethyl Substituted Homoallylamine

Abstract
An efficient asymmetric synthesis of both enantiomers of α-trifluoromethylated homoallylamine via nucleophilic allylation of trifluoroacetaldehyde SAMP- or RAMP-hydrazone, followed by benzoylation and SmI2-promoted nitrogen-nitrogen single bond cleavage is described.

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