Pyrido[4,3‐e]‐1,4‐diazepines and Pyrido[4,3‐b]‐1,5‐benzodiazepines: Synthesis and Affinity to Brain Benzodiazepine Receptors
- 1 January 1987
- journal article
- research article
- Published by Wiley in Archiv der Pharmazie
- Vol. 320 (8) , 704-710
- https://doi.org/10.1002/ardp.19873200807
Abstract
Pyrido[4,3‐e]‐1,4‐diazepines and fused tricyclic analogs thereof have been synthesized and tested for inhibition of benzodiazepine binding to receptors in various rat brain structures in comparison with standard drugs. Structure‐affinity relationships are discussed.This publication has 15 references indexed in Scilit:
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