Synthesis and structure-activity relationships of CP-122,721, a second-generation NK-1 receptor antagonist
- 3 February 1998
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 8 (3) , 281-284
- https://doi.org/10.1016/s0960-894x(98)00012-2
Abstract
No abstract availableKeywords
This publication has 3 references indexed in Scilit:
- Broad spectrum antiemetic effects of CP-122,721, a tachykinin NK1 receptor antagonist, in ferretsEuropean Journal of Pharmacology, 1996
- Discovery of an Orally Bioavailable NK1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic ActivityJournal of Medicinal Chemistry, 1995
- Discovery of a potent substance P antagonist: recognition of the key molecular determinantJournal of Medicinal Chemistry, 1992